Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15732 |
Ribociclib succinate
LEE011 琥珀酸盐,瑞博西尼琥珀酸盐,LEE011 succinate |
CDK | Cell Cycle/Checkpoint |
Ribociclib succinate (LEE011 succinate) 是一种高度特异性的CDK4/6抑制剂,IC50值分别为 10 nM 和 39 nM。它对细胞周期蛋白 B/CDK1 复合物的效力低 1000 倍。 | |||
T15731 |
Ribociclib succinate hydrate
LEE011 succinate hydrate |
CDK | Cell Cycle/Checkpoint |
Ribociclib succinate hydrate is a highly specific CDK4/6 inhibitor (IC50s: 10 nM and 39 nM, respectively). It also is over 1,000-fold less potent against the cyclin B/CDK1 complex. | |||
T15730 |
Ribociclib hydrochloride
LEE011 hydrochloride,瑞博西尼盐酸盐 |
CDK | Cell Cycle/Checkpoint |
Ribociclib hydrochloride is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively). It is over 1,000-fold less potent against the cyclin B/CDK1 complex. | |||
T6199 |
Ribociclib
瑞博西尼,LEE011 |
VEGFR; CDK | Angiogenesis; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors |
Ribociclib (LEE011) 是一种口服有效的高特异性 CDK4/6 抑制剂,IC50值分别为 10 nM 和 39 nM。 |